| 发明名称 |
SUBSTITUTED 4--PIPERIDINE-1-CARBOXYLIC ACID ESTERS AS A2AR AGONISTS |
| 摘要 |
The present invention provides substituted 4-{3-[6-amino-9-(3,4-dihydroxy-tetrahydro-furan-2-yl)-9H-purin-2-yl]-prop-2-ynyl}-piperidine-1-carboxylic acid esters and pharmaceutical compositions containing the same that are selective agonists of A2A adenosine receptors (ARs). These compounds and compositions are useful as pharmaceutical agents.
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| 申请公布号 |
US2009162292(A1) |
申请公布日期 |
2009.06.25 |
| 申请号 |
US20080338369 |
申请日期 |
2008.12.18 |
| 申请人 |
PGXHEALTH, LLC |
发明人 |
THOMPSON ROBERT D.;BEAUGLEHOLE ANTHONY;SCHMIDTMANN FRANK;RIEGER JAYSON M. |
| 分类号 |
A61K49/10;A61K31/7076;A61P37/08;C07H19/167 |
主分类号 |
A61K49/10 |
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