发明名称 |
A CYANO PIPERIDINYL-PHENIL-OXAZOLIDINONE AND USE THEREOF. |
摘要 |
The invention provides a compound of formula (I), or any of its enantiomers or mixtures thereof, or their pharmaceutically acceptable salts or solvates, for use as a medicament. The compound of formula (I) is active against Gram-positive and some Gram- negative human and veterinary pathogens with a weak monoamine oxidase (MAO) inhibitory activity. They are useful for the treatment of bacterial infections. The invention also discloses polymorphic forms of the compound (S)-N-{3-[4-(4-cyano-piperidin-1 -yl)-3-fluoro-phenyl]-2-oxo-oxazolidin-5- ylmethylj-acetamide. |
申请公布号 |
WO2009077484(A2) |
申请公布日期 |
2009.06.25 |
申请号 |
WO2008EP67503 |
申请日期 |
2008.12.15 |
申请人 |
FERRER INTERNACIONAL, S.A.;CANO, MONTSERRAT;PALOMER, ALBERT;GUGLIETTA, ANTONIO |
发明人 |
CANO, MONTSERRAT;PALOMER, ALBERT;GUGLIETTA, ANTONIO |
分类号 |
C07D413/10;A61K31/422;A61K31/454;A61P31/00 |
主分类号 |
C07D413/10 |
代理机构 |
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