摘要 |
<p>The present invention relates to process for preparing antihistaminic piperidine derivative, specifically fexofenadine and its pharmaceutically acceptable salts by using novel synthetic intermediates of following formula (I), wherein R is lower alkyl; R 2 is H, cyclopropyl, R 1 is alkyl, 4-(hydroxy-diphetiyl-methyl)-piperidin-l-yl.</p> |
申请人 |
IND-SWIFT LABORATORIES LIMITED;SRINIVASAN, CHIDAMBARAM, VENKATESWARAN;JOHAR, PERMINDER, SINGH;WADHWA, LALIT |
发明人 |
SRINIVASAN, CHIDAMBARAM, VENKATESWARAN;JOHAR, PERMINDER, SINGH;WADHWA, LALIT |