发明名称 INTERMEDIATES USEFUL FOR THE PREPARATION OF ANTIHISTAMINIC PIPERIDINE DERIVATIVE
摘要 <p>The present invention relates to process for preparing antihistaminic piperidine derivative, specifically fexofenadine and its pharmaceutically acceptable salts by using novel synthetic intermediates of following formula (I), wherein R is lower alkyl; R 2 is H, cyclopropyl, R 1 is alkyl, 4-(hydroxy-diphetiyl-methyl)-piperidin-l-yl.</p>
申请公布号 WO2007135693(A3) 申请公布日期 2009.06.11
申请号 WO2007IN00201 申请日期 2007.05.18
申请人 IND-SWIFT LABORATORIES LIMITED;SRINIVASAN, CHIDAMBARAM, VENKATESWARAN;JOHAR, PERMINDER, SINGH;WADHWA, LALIT 发明人 SRINIVASAN, CHIDAMBARAM, VENKATESWARAN;JOHAR, PERMINDER, SINGH;WADHWA, LALIT
分类号 C07D211/00;C07D211/22 主分类号 C07D211/00
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