发明名称 INDOLES WHICH ACT AS VIA RECEPTOR ANTAGONISTS.
摘要 <p>The present invention is concerned with novel indol-2-yl-carbonyl-piperidin- benzoimidazolon and indol-2-yl-carbonyl-piperidin-benzoxazolon derivatives as V1a receptor antagonists, their manufacture, pharmaceutical compositions containing them and their use as medicaments. The active compounds of the present invention are useful in the prevention and/or treatment of anxiety and depressive disorders and other diseases. Present invention comprises compounds of the general formula (I) wherein R<sup>1</sup> to R<sup>11</sup>, X and Y are as defined in the specification.</p>
申请公布号 MX2009005541(A) 申请公布日期 2009.06.05
申请号 MX20090005541 申请日期 2007.11.29
申请人 F. HOFFMANN-LA ROCHE AG. 发明人 MARK ROGERS-EVANS;RAFFAELLO MASCIADRI;PATRICK SCHNIDER.;HASANE RATNI;CATERINA BISSANTZ;CHRISTOPHE GRUNDSCHOBER
分类号 C07D401/14;A61K31/4427;A61P25/22;A61P25/24;C07D491/04 主分类号 C07D401/14
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