发明名称 |
AMORPHOUS FORM OF HETEROCYCLIC COMPOUND, SOLID DISPERSION AND MEDICINAL PREPARATION EACH COMPRISING THE SAME, AND PROCESS FOR PRODUCTION OF THE SAME |
摘要 |
<p>[PROBLEMS] The object is to improve the resorbability of a heterocyclic compound including s-triazine and a pyrimidine derivative in vitro. [MEANS FOR SOLVING PROBLEMS] Disclosed is, for example, an amorphous form of a heterocyclic compound as represented by the general formula (I) [wherein each of R's and others are as defined in the description] and including s-triazine and a pyrimidine derivative, or a hydrate, a solvate or a pharmaceutically acceptable salt of the heterocyclic compound. Also disclosed is a process for producing the amorphous form. Further disclosed are: a solid dispersion comprising the amorphous form; and a medicinal preparation comprising the solid dispersion.</p> |
申请公布号 |
WO2009066775(A1) |
申请公布日期 |
2009.05.28 |
申请号 |
WO2008JP71259 |
申请日期 |
2008.11.21 |
申请人 |
ZENYAKU KOGYO KABUSHIKIKAISHA;SUGAMA, TADAAKI;ISHIHARA, NOBUHIRO;TANAKA, YOSHIHARU;TAKAHASHI, MASAYUKI;YAGUCHI, SHINICHI;WATANABE, TETSUO |
发明人 |
SUGAMA, TADAAKI;ISHIHARA, NOBUHIRO;TANAKA, YOSHIHARU;TAKAHASHI, MASAYUKI;YAGUCHI, SHINICHI;WATANABE, TETSUO |
分类号 |
C07D403/04;A61K9/10;A61K9/14;A61K9/20;A61K9/48;A61K31/5377;A61K31/54;A61K47/38;A61P1/04;A61P1/06;A61P1/18;A61P11/00;A61P11/02;A61P11/06;A61P13/12;A61P17/00;A61P17/04;A61P17/06;A61P19/02;A61P19/08;A61P27/00;A61P27/02;A61P29/00;A61P31/04;A61P35/00;A61P35/02;A61P37/00;A61P37/02;A61P37/08;C07D413/14 |
主分类号 |
C07D403/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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