ISOMERIC PURINONES AND 1H-IMIDAZOPYRIDINONES AS PKC-THETA INHIBITORS
摘要
A chemical genus of purinones and 1H-imidazopyridinones, which are useful as PKC? inhibitors, and their methods of use are disclosed. The genus is represented by the Formula (I).
申请公布号
WO2009062059(A2)
申请公布日期
2009.05.14
申请号
WO2008US82832
申请日期
2008.11.07
申请人
PHARMACOPEIA, INC.;ROUGHTON, ANDREW;RONG, YAJING;HO, KOC-KAN;OHLMEYER, MICHAEL;DILLER, DAVID;CHAN, RAY JUI-HSIANG;LAI, GAIFA
发明人
ROUGHTON, ANDREW;RONG, YAJING;HO, KOC-KAN;OHLMEYER, MICHAEL;DILLER, DAVID;CHAN, RAY JUI-HSIANG;LAI, GAIFA