发明名称 PROCESS FOR PREPARING ACYCLIC HCV PROTEASE INHIBITORS
摘要 Disclosed are highly convergent processes for preparing compounds of formula (I), which compounds are potent active agents for the treatment of hepatitis C virus (HCV) infection: The disclosed processes use SNAr-type coupling reactions between peptidic compounds having a hydroxyproline moiety of the following formula: and halogenated or sulfonated bromoquinoline compounds.
申请公布号 US2009124809(A1) 申请公布日期 2009.05.14
申请号 US20090355157 申请日期 2009.01.16
申请人 BOEHRINGER INGELHEIM INTERNATIONAL GMBH 发明人 BUSACCA CARL ALAN;FRUTOS ROGELIO PEREZ;HADDAD NIZAR;KAPADIA SURESH R.;LORENZ JON CHARLES;SAHA ANJAN;SENANAYAKE CHRIS HUGH;WEI XUDONG
分类号 C07D417/14;A61K31/4709;C07C217/84;C07C225/22;C07D277/56;C07D417/04;C07K5/08;C07K5/083 主分类号 C07D417/14
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