4- (4-CYANOPHENYL) -1- (3-TRIFLUOROMETHYLPHENYL) -3,4, 6, 7-TETRAHYDRO-1H-PYRROLO [3, 4- D] PYRIMIDINE-2, 5-DIONE DERIVATIVES AND THEIR USE AS HUMAN NEUTROPHIL ELASTASE INHIBITORS
摘要
<p>Thirty six specific compounds having human neutrophil elastase inhibitory activity are disclosed, one of which has the structural formula (1). The compounds are useful inter alia for the treatment of inflammatory respiratory disease, and may be administered by inhalation.</p>
申请公布号
WO2009060158(A1)
申请公布日期
2009.05.14
申请号
WO2007GB04238
申请日期
2007.11.07
申请人
ARGENTA DISCOVERY LIMITED;RAY, NICHOLAS, CHARLES;FINCH, HARRY;EDWARDS, CHRISTINE;O'CONNOR, ELIZABETH;KULAGOWSKI, JANUSZ
发明人
RAY, NICHOLAS, CHARLES;FINCH, HARRY;EDWARDS, CHRISTINE;O'CONNOR, ELIZABETH;KULAGOWSKI, JANUSZ