发明名称 |
COMPOUND HAVING KINASE INGIBITOR ACTIVITY, PHARMACEUTICAL COMPOSITION CONTAINING THEREOF AND USE THEREOF FOR THE PREPARATION OF MEDICINE |
摘要 |
Selected compounds are effective for prophylaxis and treatment of diseases, such as HGF mediated diseases. The invention encompasses novel compounds, analogs, prodrugs and pharmaceutically acceptable salts thereof, pharmaceutically compositions and methods for prophylaxis and treatment of diseases and other maladies or conditions involving, cancer and the like. The subject invention also relates to processes for making such compounds as well as to intermediates useful in such processes. |
申请公布号 |
UA86614(C2) |
申请公布日期 |
2009.05.12 |
申请号 |
UA20060009287 |
申请日期 |
2005.01.24 |
申请人 |
AMGEN INC |
发明人 |
BELLON STEVEN;BOOKER SHON;BORG GEORGE;BUCHANAN JOHN L;BUCKNER WILLIAM H;CHAFFEE STUART C;CHENG YUAN;CHOQUETTE DEBORAH;DIPIETRO LUCIAN V;GERMAIN JULIE;GRACEFFA RUSSELL;HABGOOD GREGORY J;HARMANGE JEAN-CHRISTOPHE;HODOUS BRIAN L;KIM TAE-SEONG;KIM JOSEPH L;LA DANIEL;MARTIN MATTHEW W;MASSE CRAIG E;MCGOWAN DAVID C;NUNES JOSEPH J;PATEL VINOD F;POTASHMAN MICHELE;TASKER ANDREW;WEISS MATTHEW;WHITTINGTON DOUGLAS A;XI NING;XU SHIMIN |
分类号 |
A61K31/505;A61K31/47;C07D213/64;C07D213/81;C07D215/22;C07D215/233;C07D215/38;C07D215/48;C07D215/54;C07D217/24;C07D237/34;C07D239/30;C07D239/34;C07D239/46;C07D239/84;C07D239/94;C07D401/12;C07D403/12;C07D405/12;C07D407/12;C07D409/12;C07D413/12;C07D417/12;C07D471/04;C07D487/04 |
主分类号 |
A61K31/505 |
代理机构 |
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代理人 |
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