发明名称 |
THIENOPYRIMIDINES, THIENOPYRIDINES, AND PYRROLOPYRIMIDINES AS B-RAF INHIBITORS |
摘要 |
<p>The present invention relates to compounds of formula (Ia): and pharmaceutically acceptable salts thereof. The thieno[3,2-d]pyrimidine, thieno[2,3-d]pyrimidine, thieno[3,2-b]pyridine, thieno[2,3-b]pyridine, and pyrrolo[2,3-d]pyrimidine compounds selectively inhibit B-Raf kinase activity and are useful for treating disorders mediated by B-Raf kinase, and for the treatment of cancer.</p> |
申请公布号 |
WO2009059272(A1) |
申请公布日期 |
2009.05.07 |
申请号 |
WO2008US82194 |
申请日期 |
2008.11.03 |
申请人 |
WYETH;GOPALSAMY, ARIAMALA;SHI, MENGXIAO;BERGER, DAN MAARTEN;DUTIA, MINU DHANJISH;TORRES, NANCY;HOPPER, DARRIN WILLIAM |
发明人 |
GOPALSAMY, ARIAMALA;SHI, MENGXIAO;BERGER, DAN MAARTEN;DUTIA, MINU DHANJISH;TORRES, NANCY;HOPPER, DARRIN WILLIAM |
分类号 |
C07D491/04;A61K31/4365;A61K31/519;C07D495/04 |
主分类号 |
C07D491/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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