发明名称 |
HIGHLY ABSORBABLE SOLID PREPARATIONS CONTAINING SITAFLOXACINAND TARTARIC ACID |
摘要 |
A solid preparation improved in oral absorption and reduced in fluctuations of oral absorption can be obtained by incorporating an organic acid, particularly tartaric acid, in a solid preparation having, as an active ingredient, a high content of a quinolone compound, particularly sitafloxacin, having poor water solubility at pH around neutrality.
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申请公布号 |
CA2417764(C) |
申请公布日期 |
2009.05.05 |
申请号 |
CA20012417764 |
申请日期 |
2001.08.07 |
申请人 |
DAIICHI PHARMACEUTICAL CO., LTD. |
发明人 |
KOBAYASHI, HIDEO;SHIMAYA, TAKAHIRO;KIKUCHI, HIROSHI;SUZUKI, TATSUYA;ISHIDO, KOICHI;KATAOKA, KATSUO;KUROSAWA, AKIRA |
分类号 |
A61K31/4709;A61K9/20;A61K9/48;A61K31/4747;A61K47/12;A61P31/04;C07D401/04 |
主分类号 |
A61K31/4709 |
代理机构 |
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代理人 |
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主权项 |
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