| 摘要 |
THE PRESENT INVENTION RELATES TO NOVEL DERIVATIVES OF GENERAL FORMULA (I)(I)IN WHICHR3 IS A (1-6C) ALKYL, ARYL, ARYL(1-6C) ALKYL, HETEROARYL, HETEROARYL (1-6C) ALKYL,ARYL OR HETEROARYL FUSED TO A (1-10C) CYCLOALKYL, HETEROCYCLE, HETEROCYCLOALKYL, CYCLOALKYL, ADAMANTYL, POLYCYCLOALKYL, ALKENYL, ALKYNYL, CONR1 R2, COOR1, SO2 R1, C(=NH) R1 OR C(=NH)NR1 RADICAL;R5 , R6 AND R7 ARE, INDEPENDENTLY OF ONE ANOTHER, CHOSEN FROM THE FOLLOWING RADICALS: HALOGEN, CN,NO2,NH2, OH, OR8, COOH, C(O)OR8, -O-C(O)R8, NR8 R9, NHC 9O) R8, C(O)NR8 R9, NHC (S) R8, C(S)NR8 R9, SR8, S(O) R8, SO2 R8, NHSO2 R8, SO2 NR8 R9, -O-SO2 R8, -SO2-O-R8, TRIFLUOROMETHYL, TRIFULOROMETHOXY, (1-6C) ALKYL, (1-6C) ALKOXY, ARYL, ARYL (1-6C) ALKYL, HETEROARYL, HETEROARYL (1-6C) ALKYL,HETEROCYCLE, CYCLOALKYL, ALKENYL, ALKYNYL, ADAMANTYL OR POLYCYCLOALKYL.
|
