| 摘要 |
COMPOUNDS OF THE GENERAL FORMULA WHEREIN@R1IS C5, 6-CYCLOALKYL, SUNSTITUTED BY CF3, LOWER ALKYL, -(CH2)NOH, -(CH2), N-O-LOWER ALKYL, OR IS@1-BYCYCLO[2.2.1]HEPT-2-YL,@1-(7-OXA-BICYCLO[2.2.1.]HEPT-2-YL,@1-(5-EXO-HYDROXY-BICYCLO[2.2.1]HEPT-2-EXO-YL,@1-(5-EXO-HYDROXY-BICYCLO[2.2.1]HEPT-2-ENDO-YL,@OR IS 1-ADAMANTAN-1-YL;R2IS LOWER ALKYL; OR @R1 AND R2 FORM TOGETHER WITH THE N-ATOM THE GROUP 8-OXA-3-AZA-BICYCLO[3.2.1.]OCTANE;@NIS 0 OR 1;@AND PHARMACEUTICAL ACCEPTABLE ACID ADDITION SALTS THEREOF FOR THE TREATMENT OF DISEASES, RELATED TO THE A2A RECEPTOR.
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