发明名称 2,2,2-TRI-SUBSTITUTED ACETAMIDE DERIVATIVES AS GLUCOKINASE ACTIVATORS, THEIR PROCESS AND PHARMACEUTICAL APPLICATION
摘要 Compounds of the present disclosure are 2,2,2-tri-substituted acetamide derivatives of formula (I), its polymorphs, stereoisomers, prodrugs, solvates, pharmaceutically acceptable salts and formulations thereof, useful as Glucokinase activator. Processes of their preparation are also described in the disclosure. The disclosure also describes method to characterize partial glucokinase activators.
申请公布号 WO2008104994(A3) 申请公布日期 2009.04.02
申请号 WO2008IN00109 申请日期 2008.02.25
申请人 ADVINUS THERAPEUTICS PRIVATE LIMITED;MOOKHTIAR, KASIM, A.;BHUNIYA, DEBNATH;DAVE, BHAVESH;KAPKOTI, GOBIND, S.;BASU, SUJAY;CHUGH, ANITA;DE, SIDDARTHA;PALLE, VENKATA, P. 发明人 MOOKHTIAR, KASIM, A.;BHUNIYA, DEBNATH;DAVE, BHAVESH;KAPKOTI, GOBIND, S.;BASU, SUJAY;CHUGH, ANITA;DE, SIDDARTHA;PALLE, VENKATA, P.
分类号 C07D213/40;A61K31/4168;A61K31/44;A61P3/10;C07D213/75;C07D213/76;C07D213/80;C07D213/82;C07D239/42;C07D257/06;C07D261/14;C07D277/46;C07D277/82;C07D285/135;C07D417/12 主分类号 C07D213/40
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