发明名称 |
PYRAZOLO[5, 1-C] [1,2,4] TRIAZINES, METHODS FOR PREPARATION AND USE THEREOF |
摘要 |
<p>A pyrazolo[5,1-c][1,2,4]triazine compound of Formula (A): and pharmaceutically acceptable sats thereof. The multiply-substituted pyrazolo[5,1-c][1,2,4]triazine compounds of the invention selectively inhibit B-Raf kinase activity and are useful for treating disorders mediated by B-Raf kinase.</p> |
申请公布号 |
WO2009039387(A1) |
申请公布日期 |
2009.03.26 |
申请号 |
WO2008US77037 |
申请日期 |
2008.09.19 |
申请人 |
WYETH;BERGER, DAN M.;DUTIA, MINU D.;HOPPER, DARRIN W.;TORRES, NANCY |
发明人 |
BERGER, DAN M.;DUTIA, MINU D.;HOPPER, DARRIN W.;TORRES, NANCY |
分类号 |
C07D487/04;A61K31/53;A61P35/00 |
主分类号 |
C07D487/04 |
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