发明名称 |
PROPIONAMIDE DERIVATIVES USEFUL AS ANDROGEN RECEPTOR MODULATORS |
摘要 |
Compounds of formula (I) wherein R1 to R4, X and A are as defined in the claims and pharmaceutically acceptable salts and esters thereof, are disclosed. The compounds of formula (I) possess utility as tissue-selective androgen receptor modulators (SARM) and are useful in hormonal therapy, e.g. in the treatment or prevention of male hypogonadism and age-related conditions such as andropause.(I) |
申请公布号 |
UA86027(C2) |
申请公布日期 |
2009.03.25 |
申请号 |
UA20060000713 |
申请日期 |
2004.06.24 |
申请人 |
ORION CORPORATION |
发明人 |
RATILAINEN JARI;MOILANEN ANU;TOERMOKANGAS OLLI;KARJALAINEN ARJA;HUHTALA PAAVO;WOHLFAHRT GERD;KALLIO PEKKA |
分类号 |
C07C235/24;A61K31/167;A61K31/277;A61K31/395;A61P5/26;A61P15/16;C07C;C07C237/04;C07C255/54;C07C255/58;C07C275/34;C07C311/08;C07C323/20;C07D213/64;C07D213/65;C07D213/68 |
主分类号 |
C07C235/24 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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