发明名称 FLUORINE- SUBSTITUTED 2 ', 6 ' -DIMETHYL-L-TYROSINE-1, 2,3, 4-TETRAHYDR0IS0QUIN0LINE-3-CARB0XYLIC ACID PEPTIDES (DMT-TIC) FOR USE AS MYU- AND DELTA-OPIOID RECEPTOR PROBES IN
摘要 <p>Disclosed are compounds of formula (I) or pharmaceutically acceptable salts thereof: Formula (I) in which R1, R2, and R3 are described herein. Also disclosed is a pharmaceutical composition comprising at least one compound of formula (I) and a pharmaceutically acceptable carrier. Also disclosed is a method of locating a µ- and/or d-opioid receptor that is contained in a tissue or organ.</p>
申请公布号 WO2009032840(A1) 申请公布日期 2009.03.12
申请号 WO2008US75114 申请日期 2008.09.03
申请人 THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES;THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY;LAZARUS, LAWRENCE H.;BALBONI, GIANFRANCO;SALVADORI, SEVERO;CHEN, XIAOYUAN 发明人 LAZARUS, LAWRENCE H.;BALBONI, GIANFRANCO;SALVADORI, SEVERO;CHEN, XIAOYUAN
分类号 C07D217/26;A61K31/472 主分类号 C07D217/26
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