发明名称 |
METABOLITES OF THE JANUS KINASE INHIBITOR (R)-3-(4-(7H-PYRROLO[2,3-D]PYRIMIDIN-4-YL)-LH-PYRAZOL-L-YL)-3- CYCLOPENTYLPROPANENITRILE |
摘要 |
The present invention provides active metablites of 3-(4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazol-1-yl)-3-cyclopentylpropanenitrile that modulate the activity of Janus kinases and are useful in the treatment of diseases related to activity of Janus kinases including, for example, immune-related diseases, skin disorders, myeloid proliferative disorders, cancer, and other diseases. |
申请公布号 |
WO2008157207(A3) |
申请公布日期 |
2009.02.26 |
申请号 |
WO2008US66658 |
申请日期 |
2008.06.12 |
申请人 |
INCYTE CORPORATION;RODGERS, JAMES D.;ARVANITIS, ARGYRIOS G.;SHI, JACK GUOEN |
发明人 |
RODGERS, JAMES D.;ARVANITIS, ARGYRIOS G.;SHI, JACK GUOEN |
分类号 |
C07D487/04;A61K31/519 |
主分类号 |
C07D487/04 |
代理机构 |
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代理人 |
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地址 |
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