发明名称 NAPHTHYLPYRIMIDINE, NAPHTHYLPYRAZINE AND NAPHTHYLPYRIDAZINE ANALOGS AND THEIR USE AS AGONISTS OF THE WNT-BETA-CATENIN CELLULAR MESSAGING SYSTEM
摘要 <p>The present invention relates to naphthylpyrimidine analogs, methods of making naphthylpyrimidine analogs, compositions comprising a naphthylpyrimidine analog, and methods for treating canonical Wnt-[beta-symbol]-catenin cellular messaging system-related disorders comprising administering to a subject in need thereof an effective amount of a naphthylpyrimidine, naphthylpyrazine and naphthylpyridazine analog.</p>
申请公布号 WO2009026326(A1) 申请公布日期 2009.02.26
申请号 WO2008US73655 申请日期 2008.08.20
申请人 WYETH;PELLETIER, JEFFREY CLAUDE;FELIX, LUCIANA DE ARAUJO;GREEN, DANIEL MICHAEL;HAUZE, DIANE BARBARA;LUNDQUIST IV, JOSEPH THEODORE;MANN, CHARLES WILLIAM;MEHLMANN, JOHN FRANCIS;ROGERS, JR., JOHN FRANCIS;VERA, MATTHEW DOUGLAS;MOLINARI, ALBERT JOHN 发明人 PELLETIER, JEFFREY CLAUDE;FELIX, LUCIANA DE ARAUJO;GREEN, DANIEL MICHAEL;HAUZE, DIANE BARBARA;LUNDQUIST IV, JOSEPH THEODORE;MANN, CHARLES WILLIAM;MEHLMANN, JOHN FRANCIS;ROGERS, JR., JOHN FRANCIS;VERA, MATTHEW DOUGLAS;MOLINARI, ALBERT JOHN
分类号 C07D239/26;A61K31/506;A61P25/00;C07D239/34;C07D401/06;C07D403/04;C07D451/02;C07D471/04;C07D471/10;C07D487/04;C07D487/08 主分类号 C07D239/26
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