发明名称 CRYSTALLINE POLYMORPH OF BAZEDOXIFENE ACETATE
摘要 PROBLEM TO BE SOLVED: To provide a crystalline polymorph of bazedoxifene acetate exhibiting better bioavailability or better stability although the polymorphic forms occur where the same composition of matter crystallizes in a different lattice arrangement resulting in different thermodynamic properties and stability specific to the particular polymorph form. SOLUTION: The crystalline polymorph (form A) of the bazedoxifene acetate characterized according to the powder X-ray diffraction data, IR data, and DSC data, and the composition containing the crystalline polymorph are provided. The production thereof and the use thereof are also provided. COPYRIGHT: (C)2009,JPO&INPIT
申请公布号 JP2009035535(A) 申请公布日期 2009.02.19
申请号 JP20080171135 申请日期 2008.06.30
申请人 WYETH 发明人 DEMERSON CHRISTOPHER;IERA SILVIO;ALI KADUM A
分类号 C07D209/12;A61K31/55;A61K31/565;A61K31/566;A61P3/06;A61P5/30;A61P5/32;A61P9/00;A61P15/00;A61P15/12;A61P19/10;A61P35/00;C07B61/00;C07D403/12 主分类号 C07D209/12
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