发明名称 Process for the Preparation of Florfenicol
摘要 The present invention relates to a method for the preparation of Florfenicol from Fluoroamine compound, namely (1R,2S)-1-[4-(methylsulfonyl)phenyl]-2-amino-3-fluoro-1-propanol (II), by reaction with dihaloacetic acid ester in an organic solvent in presence of an inorganic base.
申请公布号 US2009043131(A1) 申请公布日期 2009.02.12
申请号 US20060922468 申请日期 2006.06.12
申请人 AUROBINDO PHARMA LIMITED 发明人 KARURU MALLIKARJUNA REDDY;GUPTA ARUN KUMAR;MEENAKSHISUNDERAM SIVAKUMARAN
分类号 C07C233/33 主分类号 C07C233/33
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