发明名称 FUSED HETEROCYCLIC DERIVATIVES USEFUL AS INHIBITORS OF THE HEPATOCYTE GROWTH FACTOR RECEPTOR
摘要 Selected compounds are effective for prophylaxis and treatment of diseases, such as HGF mediated diseases. The invention encompasses novel compounds, analogs, prodrugs and pharmaceutically acceptable salts thereof, pharmaceutical compositions and methods for prophylaxis and treatment of diseases and other maladies or conditions involving, cancer and the like. The subject invention also relates to processes for making such compounds as well as to intermediates useful in such processes.
申请公布号 WO2008008539(A3) 申请公布日期 2009.02.12
申请号 WO2007US16068 申请日期 2007.07.13
申请人 AMGEN INC.;ALBRECHT, BRIAN;BAUER, DAVID;BELLON, STEVEN;BODE, CHRISTIANE;BOOKER, SHON;BOEZIO, ALESSANDRO;CHOQUETTE, DEBORAH;D'AMICO, DERIN;HARMANGE, JEAN-CHRISTOPHE;HIRAI, SATOKO;HUNGATE, RANDALL;KIM, TAE-SEONG;LEWIS, RICHARD;LIU, LONGBIN;LOHMAN, JULIA;NORMAN, MARK;POTASHMAN, MICHELE;SIEGMUND, AARON;SPRINGER, STEPHANIE;STEC, MARKIAN;XI, NING;YANG, KEVIN 发明人 ALBRECHT, BRIAN;BAUER, DAVID;BELLON, STEVEN;BODE, CHRISTIANE;BOOKER, SHON;BOEZIO, ALESSANDRO;CHOQUETTE, DEBORAH;D'AMICO, DERIN;HARMANGE, JEAN-CHRISTOPHE;HIRAI, SATOKO;HUNGATE, RANDALL;KIM, TAE-SEONG;LEWIS, RICHARD;LIU, LONGBIN;LOHMAN, JULIA;NORMAN, MARK;POTASHMAN, MICHELE;SIEGMUND, AARON;SPRINGER, STEPHANIE;STEC, MARKIAN;XI, NING;YANG, KEVIN
分类号 C07D471/04;A61K31/437;A61K31/5025;A61K31/52;A61P35/00;C07D473/34;C07D487/04 主分类号 C07D471/04
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