发明名称 IMIDAZOLOPYRIMIDINE ANALOGS AND THEIR USE AS PI3 KINASE AND MTOR INHIBITORS
摘要 The present invention relates to Imidazolopyrimidine Analogs, of Formula Ib methods of making Imidazolopyrimidine Analogs, compositions comprising an Imidazolopyrimidine Analog, and methods fot treating ot preventing a PI3K-related disorder comprising administering to a subject in need thereof an effective amount of an Imidazolopyrimidine Analog. The invention also relates to methods for treating or preventing mTOR -related disorders comprising administering to a subject in need thereof an effective amount of an Imidazolopyrimidine Analog.
申请公布号 WO2008116129(A3) 申请公布日期 2009.02.12
申请号 WO2008US57771 申请日期 2008.03.21
申请人 WYETH;BURSAVICH, MATTHEW, GREGORY;VENKATESAN, ARANAPAKAM, MUDUMBAI;NOWAK, PAWEL, WOJCIECH;LOMBARDI, SABRINA;GILBERT, ADAM, MATTHEW;DEHNHARDT, CHRISTOPH, MARTIN;DOS SANTOS, OSVALDO;DELOS SANTOS, EFREN, GUILLERMO;BROOIJMANS, NATASJA;AYRAL-KALOUSTIAN, SEMIRAMIS;CHEN, ZECHENG;VERHEIJEN, JEROEN, CUNERA;KAPLAN, JOSHUA;ZASK, ARIE 发明人 BURSAVICH, MATTHEW, GREGORY;VENKATESAN, ARANAPAKAM, MUDUMBAI;NOWAK, PAWEL, WOJCIECH;LOMBARDI, SABRINA;GILBERT, ADAM, MATTHEW;DEHNHARDT, CHRISTOPH, MARTIN;DOS SANTOS, OSVALDO;DELOS SANTOS, EFREN, GUILLERMO;BROOIJMANS, NATASJA;AYRAL-KALOUSTIAN, SEMIRAMIS;CHEN, ZECHENG;VERHEIJEN, JEROEN, CUNERA;KAPLAN, JOSHUA;ZASK, ARIE
分类号 C07D473/34;A61K31/52;A61P35/00 主分类号 C07D473/34
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