发明名称 |
PALIPERIDONE DERIVATIVES |
摘要 |
<p>A compound of formula (1) is useful as a pharmaceutical and as an intermediate in making paliperidone, wherein Y is an acid-sensitive group of the formula (A') in which X represents an oxygen atom, a sulfur atom, or an -NH- group; Z represents a C2-C7 alkylene bridge; and R represents hydrogen or a C1-C4 alkyl group.</p> |
申请公布号 |
WO2009015828(A1) |
申请公布日期 |
2009.02.05 |
申请号 |
WO2008EP06122 |
申请日期 |
2008.07.25 |
申请人 |
SYNTHON B.V.;BARTL, JIRI;PICHA, FRANTISEK |
发明人 |
BARTL, JIRI;PICHA, FRANTISEK |
分类号 |
C07D471/04;A61K31/519;A61P25/18 |
主分类号 |
C07D471/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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