发明名称 |
NEW CRYSTALLINE FORMS OF 2 -HYDROXY- 3- [5- (MORPHOLIN- 4- YLMETHYL) PYRIDIN-2-YL] IH- INDOLE- 5 -CARBONITRILE CITRATE |
摘要 |
<p>The present invention relates to new crystalline forms of 2-hydroxy-3-[5-(morpholin-4- ylmethyl)pyridin-2-yl]1H-indole-5-carbonitrile citrate, a Form D and a Form E, respectively, a process for their preparations, pharmaceutical formulations containing said compounds and to the use of said active compounds in therapy, and particularly to GSK3 related conditions and disorders.</p> |
申请公布号 |
WO2009017452(A1) |
申请公布日期 |
2009.02.05 |
申请号 |
WO2008SE50895 |
申请日期 |
2008.07.29 |
申请人 |
PROFIR, VERONICA;SEBHATU, TESFAI;TJERNELD, ERICA;ASTRAZENECA AB;ERIKSON, ANDERS |
发明人 |
ERIKSON, ANDERS;PROFIR, VERONICA;SEBHATU, TESFAI;TJERNELD, ERICA |
分类号 |
C07D413/14;A61K31/5377;A61P3/10;A61P19/04;A61P19/10;A61P25/16;A61P25/18;A61P25/28;A61P29/00 |
主分类号 |
C07D413/14 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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