发明名称 PROCESS FOR THE PREPARATION OF CYCLIC SPIROPIPERIDINES
摘要 <p>The present invention relates to new processes for the preparation of compounds of formula I, especially the compound 2-{2-Chloro-5-{[(2S)-3-(5-chloro-1'H,3H-spiro[1- benzofuran-2,4'-piperidin]-1'-yl)-2-hydroxypropyl]oxy}-4-5 [(methylamino)carbonyl]phenoxy}-2-methylpropanoic acid and to new intermediates useful in the preparation thereof.</p>
申请公布号 WO2009011654(A1) 申请公布日期 2009.01.22
申请号 WO2008SE50877 申请日期 2008.07.16
申请人 ASTRAZENECA AB;IVANOVA, SVETLANA;KAVITAKE, SANTOSH;KUMAR, SYTHANA SURESH;LINGESHA, SIDDA;MENSONIDES-HARSEMA, MARGUERITE;MERIFIELD, ERIC;PAVEY, JOHN;KUMAR, VINOD;ENNIS, DAVID 发明人 IVANOVA, SVETLANA;KAVITAKE, SANTOSH;KUMAR, SYTHANA SURESH;LINGESHA, SIDDA;MENSONIDES-HARSEMA, MARGUERITE;MERIFIELD, ERIC;PAVEY, JOHN;KUMAR, VINOD;ENNIS, DAVID
分类号 C07D491/107;C07C69/92;C07C235/60;C07D303/24 主分类号 C07D491/107
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