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发明名称
胺基-杂环化合物
摘要
本发明提供式(I)之PDE9-抑制性化合物,#P 097117227P01.bmp及其药学上可接受之盐类,其中R、R#sB!1#eB!、R#sB!2#eB!以及R#sB!3#eB!系如同在此所定义。含有式I化合物之药学组成物及其于治疗诸如阿兹海默症及精神分裂之神经退化性疾病及认知疾病的用途亦被提供。
申请公布号
TW200902015
申请公布日期
2009.01.16
申请号
TW097117227
申请日期
2008.05.09
申请人
辉瑞股份有限公司
发明人
威赫斯特 派克R;浦鲁克斯弗朗西 卡洛琳
分类号
A61K31/519(2006.01);C07D487/04(2006.01);A61P25/00(2006.01);A61P25/28(2006.01)
主分类号
A61K31/519(2006.01)
代理机构
代理人
恽轶群;陈文郎
主权项
地址
美国
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