发明名称 Bis-2-difluoro-pyrrolo[2,1-C][1,4]benzodiazepine dimers
摘要 The present invention provides a novel bis 2-difluoro pyrrolo[2,1-c][1,4]benzodiazepine of formula VII wherein, n is 3 to 10. novel bis 2-difluoro pyrrolo[2,1-c][1,4]benzodiazepine of formula VII exhibits biding affinity with calf thymus (CT) DNA at a molar ratio of 1:5 in aqueous sodium phosphate buffer at pH of about 7.00. The present invention further provides a process for the preparation of novel bis 2-difluoro pyrrolo[2,1-c][1,4]benzodiazepine of formula VII.
申请公布号 US7476664(B2) 申请公布日期 2009.01.13
申请号 US20070715592 申请日期 2007.03.07
申请人 KAMAL AHMED;REDDY DEPATLA RAJASEKHAR;RAJENDAR RAJENDAR 发明人 KAMAL AHMED;REDDY DEPATLA RAJASEKHAR;RAJENDAR RAJENDAR
分类号 C07D405/14;A61K31/551;A61P25/06 主分类号 C07D405/14
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