发明名称 High-concentration lidocaine compositions and methods for their preparation
摘要 A composition comprising lidocaine-containing liposomes wherein the weight concentration of lidocaine in said composition is greater than 10%. The composition is prepared by mixing water with an oil phase comprising lidocaine, a C14-C20 alcohol, an alkyl ester of a fatty acid, propylene glycol, and a polyalkyl stearate. The non-aqueous phase may also include a phospholipid such as phosphatidyl choline.
申请公布号 US7476400(B2) 申请公布日期 2009.01.13
申请号 US20020290983 申请日期 2002.11.08
申请人 FERNDALE IP, INC. 发明人 PATEL PRAVIN M.
分类号 A61K9/127;A61K9/00;A61K31/165;A61K31/167;A61K47/10;A61K47/14;A61K47/22;A61K47/24;A61K47/34;A61P23/02 主分类号 A61K9/127
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