发明名称 |
NOVEL ARYLAMIDINE DERIVATIVE, SALT THEREOF ,AND ANTIFUNGAL CONTAINING THESE |
摘要 |
An arylamidine derivative represented by the general formula (wherein R 1 represents optionally protected or substituted amidino; and R 2 and R 3 are the same or different and each represents hydrogen or halogeno) or a salt of the derivative. The derivative and salt have potent activity against fungi including ones having tolerance to azole type drugs and further have high safety and excellent properties in a repeated dose toxicity test. They are hence useful as an excellent antifungal. |
申请公布号 |
ZA200700806(B) |
申请公布日期 |
2008.12.31 |
申请号 |
ZA20070000806 |
申请日期 |
2007.01.29 |
申请人 |
TOYAMA CHEMICAL CO . LTD |
发明人 |
HAYASHI KAZUYA;KUNITANI KAZUTO;UEHARA SAYURI;MORITA TEIICHI |
分类号 |
C07D;A61K;A61P |
主分类号 |
C07D |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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