发明名称 NOVEL POLYHYDROXYLATED COMPOUNDS AS FATTY ACID SYNTHASE (FASN) INHIBITORS
摘要 The present invention relates to new polyhydroxylated compounds and, in particular, to its activity as fatty acid synthase (FASN) inhibitors and to their use for the treatment of pathological states for which an inhibitor of this enzyme is indicated. The invention further relate to pharmaceutical compositions containing them and to a process for the preparation of such compounds.
申请公布号 WO2009000864(A1) 申请公布日期 2008.12.31
申请号 WO2008EP58099 申请日期 2008.06.25
申请人 FUNDACIO PRIVADA INSTITUT D'INVESTIGACIO BIOMEDICA DE GIRONA DR. JOSEP TRUETA;UNIVERSIDAD COMPLUTENSE DE MADRID;COLOMER BOSCH, RAMON;PUIG MIQUEL, TERESA;BRUNET VIDAL, JOAN;LOPEZ RODRIGUEZ, MARIA LUZ;BENHAMU SALAMA, BELLINDA;ORTEGA GUTIERREZ, SILVIA;TURRADO GARCIA, CARLOS 发明人 COLOMER BOSCH, RAMON;PUIG MIQUEL, TERESA;BRUNET VIDAL, JOAN;LOPEZ RODRIGUEZ, MARIA LUZ;BENHAMU SALAMA, BELLINDA;ORTEGA GUTIERREZ, SILVIA;TURRADO GARCIA, CARLOS
分类号 C07C69/94;C07D213/79 主分类号 C07C69/94
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