发明名称 7-Pyrazolylbenzazepines Having Affinity For D3 Receptor
摘要 Compounds of formula (I) or a salt thereof are disclosed: wherein R1 is pyrazolyl substituted by two or three substituents independently selected from halogen, C1-4alkyl and haloC1-4alkyl; R2 is hydrogen or methyl; and R3 is quinolinyl, oxazolyl or phenyl, each of which is optionally substituted by one or two halogen, C1-4alkyl or haloC1-4alkyl. Processes for preparation and uses of the compounds in medicine, for example for the treatment of schizophrenia or drug dependency, are also disclosed.
申请公布号 US2008312213(A1) 申请公布日期 2008.12.18
申请号 US20050570623 申请日期 2005.06.17
申请人 GLAXO GROUP LIMITED 发明人 HAMPRECHT DIETER;MICHELI FABRIZIO;TARSI LUCA;TEDESCO GIOVANNA
分类号 A61K31/55;C07D401/14;C07D403/14;C07D413/14 主分类号 A61K31/55
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