发明名称 QUINOLINONE DERIVATIVES AS PARP AND TANK INHIBITORS
摘要 The present invention provides compounds of Formula (I), their use as PARP inhibitors as well as pharmaceutical compositions comprising said compounds, wherein R<SUP>1</SUP>, R<SUP>2</SUP>, R<SUP>3</SUP>, R<SUP>4</SUP>, R<SUP>5</SUP>, R<SUP>6</SUP>, R<SUP>7</SUP>, n, m and X have defined meanings.
申请公布号 WO2008107478(A8) 申请公布日期 2008.10.23
申请号 WO2008EP52764 申请日期 2008.03.07
申请人 JANSSEN PHARMACEUTICA NV;VIALARD, JORGE EDUARDO;ANGIBAUD, PATRICK RENE;MEVELLEC, LAURENCE ANNE;MEYER, CHRISTOPHE;FREYNE, EDDY JEAN EDGARD;PILATTE, ISABELLE NOELLE CONSTANCE;ROUX, BRUNO;PASQUIER, ELISABETH THERESE JEANNE;BOURDREZ, XAVIER MARC;ADELINET, CHRISTOPHE DENIS;MARCONNET-DECRANE, LAURENCE FRANCOISE BERNADETTE;MACRITCHIE, JACQUELINE ANNE;DUFFY, JAMES EDWARD STEWART;OWENS, ANDREW PATE;STORCK, PIERRE-HENRI;PONCELET, VIRGINIE SOPHIE 发明人 VIALARD, JORGE EDUARDO;ANGIBAUD, PATRICK RENE;MEVELLEC, LAURENCE ANNE;MEYER, CHRISTOPHE;FREYNE, EDDY JEAN EDGARD;PILATTE, ISABELLE NOELLE CONSTANCE;ROUX, BRUNO;PASQUIER, ELISABETH THERESE JEANNE;BOURDREZ, XAVIER MARC;ADELINET, CHRISTOPHE DENIS;MARCONNET-DECRANE, LAURENCE FRANCOISE BERNADETTE;MACRITCHIE, JACQUELINE ANNE;DUFFY, JAMES EDWARD STEWART;OWENS, ANDREW PATE;STORCK, PIERRE-HENRI;PONCELET, VIRGINIE SOPHIE
分类号 C07D215/22;A61K31/4704 主分类号 C07D215/22
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