发明名称 Pyrazole Derivatives Having Tyrosine Kinase Activity
摘要 Compounds of the formula (I), in which R, X, R<SUP>1</SUP>, R<SUP>2</SUP>, R<SUP>3 </SUP>and R<SUP>4 </SUP>have the meanings indicated in Claim ( 1 ), are inhibitors of tyrosine kinases, in particular TIE-2, and Raf kinases and can be employed, inter alia, for the treatment of tumours.
申请公布号 US2008207647(A1) 申请公布日期 2008.08.28
申请号 US20060063020 申请日期 2006.07.24
申请人 MERCK PATENT GMBH 发明人 HOELZEMANN GUENTER;CRASSIER HELENE;RAUTENBERG WILFRIED
分类号 A61K31/52;A61K31/4178;A61K31/519;A61P19/00;A61P27/00;A61P29/00;A61P35/00;C07D403/12;C07D471/04;C07D487/04 主分类号 A61K31/52
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