PROCESS FOR THE PREPARATION OF (2R,3S)-3-PHENYLISOSERINE METHYL ESTER ACETATE SALT
摘要
<p>A process for the enantioselective preparation of (2R,3S)-3-phenylisoserine methyl ester acetate salt of formula (I) which is an useful building block for the synthesis of taxane derivatives. The process involves the resolution of racemic threo-phenylisoserine amide and its conversion into (I).</p>
申请公布号
WO2008101608(A1)
申请公布日期
2008.08.28
申请号
WO2008EP01015
申请日期
2008.02.11
申请人
INDENA S.P.A.;CICERI, DANIELE;GABETTA, BRUNO;VIGNOLA, NICOLA;MITZEL, FRIEDER;WEBER, BEAT, T.
发明人
CICERI, DANIELE;GABETTA, BRUNO;VIGNOLA, NICOLA;MITZEL, FRIEDER;WEBER, BEAT, T.
