发明名称 |
NOVEL METHOD FOR SYNTHESISING DERIVATIVES OF (2S, 3aS, 7aS)-1-[(S)-ALANYL]-OCTAHYDRO-1H-INDOLE-2-CARBOXYLIC ACID AND THE USE THEREOF FOR PERINDOPRIL SYNTHESIS |
摘要 |
The invention relates to a method for synthesising compounds of the formula (I)wherein Ris a hydrogen atom or an alkyl or benzyl group, and Ris amine function protecting group representing tert-butoxycarbonyl.The use of said compounds for synthesising perindopril and the pharmaceutically acceptable salts thereof is also disclosed. |
申请公布号 |
EA009062(B1) |
申请公布日期 |
2007.10.26 |
申请号 |
EA20050001257 |
申请日期 |
2004.02.27 |
申请人 |
LES LABORATOIRES SERVIER |
发明人 |
DUBUFFET THIERRY;LANGLOIS PASCAL |
分类号 |
C07K5/06;C07D209/42;C07K5/02 |
主分类号 |
C07K5/06 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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