发明名称 NOVEL METHOD FOR SYNTHESISING DERIVATIVES OF (2S, 3aS, 7aS)-1-[(S)-ALANYL]-OCTAHYDRO-1H-INDOLE-2-CARBOXYLIC ACID AND THE USE THEREOF FOR PERINDOPRIL SYNTHESIS
摘要 The invention relates to a method for synthesising compounds of the formula (I)wherein Ris a hydrogen atom or an alkyl or benzyl group, and Ris amine function protecting group representing tert-butoxycarbonyl.The use of said compounds for synthesising perindopril and the pharmaceutically acceptable salts thereof is also disclosed.
申请公布号 EA009062(B1) 申请公布日期 2007.10.26
申请号 EA20050001257 申请日期 2004.02.27
申请人 LES LABORATOIRES SERVIER 发明人 DUBUFFET THIERRY;LANGLOIS PASCAL
分类号 C07K5/06;C07D209/42;C07K5/02 主分类号 C07K5/06
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