| 摘要 |
The invention relates to 6-phenyl-7-amino-triazolopyrimidines of formula (I), wherein the substituents have the following designations: R1 represents hydrogen, alkyl, halogenalkyl, cycloalkyl, halogencycloalkyl, alkenyl, halogenalkenyl, cycloalkenyl, halogencycloalkenyl, alkinyl, halogenalkinyl or phenyl, naphthyl, or a five-membered or six-membered saturated, partially unsaturated or aromatic heteroycle, containing between one and four heteroatoms from the group containing O, N or S; R2 represents alkyl, halogenalkyl, cycloalkyl, halogencycloalkyl, alkenyl, halogenalkenyl, cycloalkenyl, halogencycloalkenyl, alkinyl, halogenalkinyl or phenyl, naphthyl, or a five-membered or six-membered saturated, partially unsaturated or aromatic heterocycle, containing between one and four heteroatoms from the group containing O, N or S; R3,R4,R5, R6,R7 represent hydrogen or one of the groups cited for R2, R4 also being able to form a five-membered or six-membered saturated or unsaturated ring with R3 or R 6, that can contain, in addition to carbon atoms and as a ring member, between one and three other heteroatoms from the group containing O, N and S; R2 and R3, R4 and R 5, and R6 and R7 can respectively form, in order to form spiro groups, a C2-C5 alkylene, alkenylene, or alkinylene chain, which can be broken by between one and three heteroatoms from the group containing O, N and S; p represents 0 or 1; L represents halogen, alkyl, halogenalkyl, alkoxy, cyano, nitro, amino, alkylamino, dialkylamino, alkylcarbonylamino, C(O)-R, S(O)n-R; where n represents 0, 1 or 2; R represents hydrogen, alkyl, halogenalkyl, alkoxy, alkenyloxy, alkinyloxy, amino, alkylamino, dialkylamino; m represents 1, 2, 3, 4 or 5; X represents halogen, cyano, alkyl, alkoxy, alkenyloxy, alkinyloxy or halogenalkoxy, Y represents oxygen or sulphur; Z represents hydrogen, alkyl, halogenalkyl, cycloalkyl, alkylcarbonyl, cycloalkylcarbonyl, alkenyl, halogenalkenyl, cycloalkenyl, alkinyl, halogenalkinyl, phenyl, naphthyl, a five-membered to ten-membered saturated, partially unsaturated or aromatic heterocycle, containing between one and four heteroatoms from the group containing O, N and S; or Z can also form, with R4 or R6, a five-membered or six-membered ring that can contain, in addition to carbon atoms and Y, one or two other heteroatoms from the group containing O, N and S, as a ring member; the groups R1 to R7, Z and R being able to be substituted according to the description. The invention also relates to methods for producing said compounds, to agents containing the same, and to the use thereof for controlling plant pathogenic fungi.
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