发明名称 PROCESS FOR PRODUCTION OF CARBAPENEM DERIVATIVE AND CRYSTALLINE INTERMEDIATE THEREFOR
摘要 Disclosed is an intermediate for the synthesis of a carbapenem which is advantageous for the industrial production of the carbapenem. A process for producing a compound (I) or a pharmaceutically acceptable salt or solvate thereof or a crystal thereof, comprising reacting a compound (III) with a compound (IV) in the presence of a secondary amine; a crystal of a benzyl alcohol-solvated form of the compound (I) or the like; a method for deprotecting the compound (I) by using a Pd catalyst; and a crystal of the compound (IV) or the like.
申请公布号 KR20070104594(A) 申请公布日期 2007.10.26
申请号 KR20077018449 申请日期 2007.08.10
申请人 SHIONOGI & CO., LTD. 发明人 UENAKA MASAAKI;HOZUMI YASUYUKI;NOGUCHI KOUICHI;KOMURASAKI TADAFUMI
分类号 C07D477/20;C07D477/00 主分类号 C07D477/20
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