发明名称 Substituted azaindoles as inhibitors of protein kinases, and process for their preparation
摘要 Physiologically active substituted azaindole compounds of general formula (I): compositions containing such compounds; their prodrugs, and pharmaceutically acceptable salts and solvates of such compounds and their prodrugs are disclosed, wherein the variables shown in formula (I) are as defined in the specification. Such compounds and compositions have valuable pharmaceutical properties, in particular the ability to inhibit kinases, whereby these compounds are suitable for use in the treatment of disease states capable of being modulated by the inhibition of the protein kinases.
申请公布号 NZ529205(A) 申请公布日期 2006.04.28
申请号 NZ20020529205 申请日期 2002.06.20
申请人 AVENTIS PHARMA LIMITED 发明人 COX, PAUL JOSEPH;MAJID, TAHIR NADEEM;LAI, JUSTINE YEUN QUAI;MORLEY, ANDREW;AMENDOLA, SHELLEY;DEPRETS, STEPHANIE DANIELE;EDLIN, CHRIS;GARDNER, CHARLES J;KOMINOS, DOROTHEA;PEDGRIFT, BRIAN LESLIE;HALLEY, FRANK;GILLESPY, TIMOTHY ALAN;EDWARDS, MICHAEL;CLERC, FRANCOIS FREDERIC;NEMECEK, CONCEPTION;HOUILLE, OLIVIER;DAMOUR, DOMINIQUE;BOUCHARD, HERVE;BEZARD, DANIEL;CARREZ, CHANTAL
分类号 A61K;A61K31/437;A61K31/4709;A61K31/4725;A61K31/496;A61K31/4985;A61K31/5355;A61K31/5377;A61K31/541;A61P;A61P9/00;A61P11/00;A61P11/02;A61P11/06;A61P13/08;A61P17/00;A61P17/02;A61P17/06;A61P19/02;A61P27/14;A61P29/00;A61P35/00;A61P37/08;A61P43/00;C07D;C07D471/04;C07D487/04;C07D519/00;(IPC1-7):C07D471/04;A61K31/498 主分类号 A61K
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