发明名称 PROCESS FOR THE PREPARATION OF 6,6-DIMETHYL-3-AZABICYCLO- [3.1.0]- HEXANE COMPOUNDS UTILIZING BISULFITE INTERMEDIATE
摘要 The present invention provides for a process for preparing 6,6-Dimethyl-3 -aza-bicyclo[3.1.0]hexane-2-sulfonate, an intermediateuseful in the efficien t preparation of (1R, 2S, 5S)-methyl 6,6-dimethyl-3-azabicyclo[3,1,0]hexane- 2-carboxylic acid and esters and salts thereof, processes for preparing (1R, 2S, 5S)-methyl 6,6-dimethyl-3-azabicyclo[3,1,0]hexane-2-carboxylic acid and esters and salts thereof from the sulfonate intermediate and processes for preparing 6,6-Dimethyl-3-aza-bicyclo[3.1.0]hexane-2-sulfonate.
申请公布号 CA2672701(A1) 申请公布日期 2008.07.10
申请号 CA20072672701 申请日期 2007.12.18
申请人 SCHERING CORPORATION 发明人 DEMONCHAUX, PATRICE;BERRANGER, THIERRY
分类号 C07D209/54 主分类号 C07D209/54
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