| 发明名称 |
3-CARBAMOYL-2-PYRIDONE DERIVATIVE |
| 摘要 |
<P>PROBLEM TO BE SOLVED: To provide a 3-carbamoyl-2-pyridone derivative having a cannabinoid receptor agonist action, and to provide a pharmaceutical composition containing the compound as an active ingredient. <P>SOLUTION: The 3-carbamoyl-2-pyridone derivative is represented by general formula (I) [R<SP>1</SP>is a 1 to 8C alkyl, or the like; R<SP>2</SP>is a 1 to 6C alkyl; R<SP>3</SP>is a 1 to 6C alkyl or the like, or R<SP>2</SP>and R<SP>3</SP>may together form a five- to ten-membered non-aromatic carbon ring; R<SP>4</SP>is H or the like; G is a group represented by formula (A) (R<SP>5</SP>is H or the like; X<SP>1</SP>is a single bond or the like; X<SP>2</SP>is a 1 to 8C alkylene or the like; X<SP>3</SP>is a single bond or the like)], and its pharmaceutically acceptable salt or their solvates are disclosed. <P>COPYRIGHT: (C)2008,JPO&INPIT |
| 申请公布号 |
JP2008156366(A) |
申请公布日期 |
2008.07.10 |
| 申请号 |
JP20080010009 |
申请日期 |
2008.01.21 |
| 申请人 |
SHIONOGI & CO LTD |
发明人 |
ISHIZUKA NATSUKI;SASAYA TAKASHI;HIRAMATSU YOSHIHARU;INAGAKI MASANAO;ODAN MASAHIDE;HASHIZUME HIROSHI;MITSUMORI SUSUMU;FUJII YASUHIKO;FUKUI KIICHI;WATABE HIDEAKI;SATO JUN |
| 分类号 |
C07D213/82;A61K31/435;A61K31/4365;A61K31/444;A61K31/4545;A61K31/455;A61K31/496;A61K31/506;A61K31/5377;A61K31/55;A61P17/00;A61P17/04;A61P43/00;C07D221/04;C07D401/12;C07D405/12;C07D409/12;C07D413/12;C07D417/12;C07D417/14;C07D495/04 |
主分类号 |
C07D213/82 |
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