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发明名称
新颖咯酮衍生物及含有其之药学组成物
摘要
本发明提供一种式(I)所示之化合物、制药上可接受之盐或是该等之溶剂合物,而作为P2X#sB!3#eB!及/或P2X#sB!2/3#eB!拮抗剂甚为有用,即:#P 097111332P01.bmp式中,R#sP!1#eP!、R#sP!2#eP!、R#sP!3#eP!、Z#sP!1#eP!、Z#sP!2#eP!、R#sP!a#eP!、R#sP!b#eP!、q、A及n系如说明书中所定义者。
申请公布号
TW200843739
申请公布日期
2008.11.16
申请号
TW097111332
申请日期
2008.03.28
申请人
野义制药股份有限公司 SHIONOGI &
发明人
甲斐浩幸;筱原俊次;龟山贵之
分类号
A61K31/407(2006.01);A61K31/4427(2006.01);A61K31/4162(2006.01);C07D487/02(2006.01);C07D401/10(2006.01);C07D413/10(2006.01);C07D417/04(2006.01);C07D417/14(2006.01);C07D403/10(2006.01)
主分类号
A61K31/407(2006.01)
代理机构
代理人
恽轶群;陈文郎
主权项
地址
日本
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