发明名称 Glucopyranosyloxy benzylbenzene derivatives, medicinal compositions containing the same and intermediates for the preparation of the derivatives
摘要 The present invention relates to glucopyranosyloxybenzylbenzene derivatives represented by the general formula: wherein R1 represents a hydrogen atom or a hydroxy(lower alkyl) group; and R2 represents a lower alkyl group, a lower alkoxy group, a lower alkylthio group, a hydroxy(lower alkyl) group, a hydroxy(lower alkoxy) group, a hydroxy(lower alkylthio) group etc., and salts thereof, which have an excellent inhibitory activity in human SGLT2 and are useful as agents for the prevention or treatment of diabetes, obesity etc., and intermediates thereof.
申请公布号 US7465712(B2) 申请公布日期 2008.12.16
申请号 US20020221843 申请日期 2002.12.30
申请人 KISSEI PHARMACEUTICAL CO., LTD. 发明人 FUJIKURA HIDEKI;FUSHIMI NOBUHIKO;NISHIMURA TOSHIHIRO;TATANI KAZUYA
分类号 A01N43/04;A61K31/70;A61K31/7034;A61P3/04;A61P3/10;A61P43/00;C07C39/04;C07C69/16;C07C69/18;C07C69/78;C07C323/18;C07H15/203 主分类号 A01N43/04
代理机构 代理人
主权项
地址