发明名称 Substituted pyrrolo[2.3-B]pyridines
摘要 Compounds represented by Formula (I): or stereoisomers or pharmaceutically acceptable salts thereof, are inhibitors of least two of the Abl, Aurora-A, Blk, c-Raf, cSRC, Src, PRK2, FGFR3, Flt3, Lck, Mek1, PDK-1, GSK3beta, EGFR, p70S6K, BMX, SGK, CaMKII, Tie-2, IGF-1R, Ron, Ret, and KDR kinases in animals, including humans, for the treatment and/or prevention of various diseases and conditions such as cancer.
申请公布号 US7465726(B2) 申请公布日期 2008.12.16
申请号 US20050194158 申请日期 2005.08.01
申请人 OSI PHARMACEUTICALS, INC. 发明人 AHMED SALEH;BARBA OSCAR;BLOXHAM JASON;DAWSON GRAHAM;GATTRELL WILLIAM;KITCHIN JOHN;PEGG NEIL ANTHONY;SABA IMAAD;SADIQ SHAZIA;SAMBROOK SMITH COLIN PETER;SMYTH DON;STEINIG AMO G.;WILKES ROBIN;PANICKER BIJOY;TAVARES PAULA;COX MATTHEW;LI AN-HU;DONG HANQING;MA LIFU;FOREMAN KENNETH ('KEN');WENG QINGHUA ('FELIX');STOLZ KATHRYN
分类号 A61K31/437;A61K31/04;A61K31/496;A61K31/519;A61K31/5355;A61K31/541;A61K31/551;A61K31/5513;C07D223/04;C07D241/04;C07D243/08;C07D413/06;C07D413/08;C07D413/10;C07D413/12;C07D413/14;C07D417/06;C07D417/14;C07D471/04;C07D487/04 主分类号 A61K31/437
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