摘要 |
Disclosed is a pyrimidodiazepinone derivative represented by the general formula (I) below, or a pharmaceutically acceptable salt thereof. (I) (In the formula, n represents 1 or 2; Z represents a hydrogen atom or the like; R1 and R2 may be the same or different and represent a hydrogen atom or the like; A represents a bond, a (CH2)m group (wherein m represents an integer of 1-4), an optionally substituted phenylene, an optionally substituted pyridinediyl, or a C=O group; R3 represents a hydrogen atom, an optionally substituted lower alkyl group or the like; and R4 represents a hydrogen atom or the like.)
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申请人 |
KYOWA HAKKO KIRIN CO., LTD.;OTSUBO, NOBUMASA;TSUKUMO, YUKIHITO;UCHIDA, KENJI;MATSUMOTO, YUICHI;IIDA, KYOICHIRO;TAKADA, HIDENORI;TAKIZAWA, FUMITAKE;ARAI, HITOSHI;OKAZAKI, SHUKO;IMAIZUMI, TAKAMICHI |
发明人 |
OTSUBO, NOBUMASA;TSUKUMO, YUKIHITO;UCHIDA, KENJI;MATSUMOTO, YUICHI;IIDA, KYOICHIRO;TAKADA, HIDENORI;TAKIZAWA, FUMITAKE;ARAI, HITOSHI;OKAZAKI, SHUKO;IMAIZUMI, TAKAMICHI |