发明名称 3H-QUINAZOLIN-4-ON DERIVATIVES AND MEDICATION, POSSESSING PROPERTIES OF SPECIFIC MONOAMINOOXIDASE B INHIBITOR
摘要 FIELD: chemistry. ^ SUBSTANCE: in compound of formula I R1 is -(CH2)n-CO-NR5R6; -(CH2)n-COOR7; -(CH2)n- NR5R6; -(CH2)n-CN; -(CH2)n-OR8 or phenyl, which is unsubstituted or substituted with from one to three substituents, selected from halogen; R2 is hydrogen; R3 is hydrogen, (C1-C6)-alkyl, (C3-C6)-cycloalkyl or benzyl; R4 is halogen; R5 and R6 are hydrogen; R7 is hydrogen or C1-C6-alkyl; R8 is C1-C6-alkyl; m is 1, 2 or 3; and n is 0, 1 or 2. ^ EFFECT: increase of composition and treatment method efficiency. ^ 5 cl, 2 dwg, 27 ex
申请公布号 RU2340604(C2) 申请公布日期 2008.12.10
申请号 RU20050121908 申请日期 2003.12.08
申请人 F.KHOFFMANN-LJA ROSH AG 发明人 RODRIGES-SARM'ENTO ROSA-MARIJA;TOMAS EHNDR'JU UILL'JAM;VILER RENE
分类号 C07D239/91;A61K31/517;A61P25/28;C07D239/00;C07D239/90 主分类号 C07D239/91
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