| 摘要 |
The invention relates to the triazolopyridine carboxamide derivatives and triazolopyrimidine carboxamide derivatives of general formula (I) in which: A and X are, independently of one another, a nitrogen atom or a CH group; R1 is an NR3R4 group, in which R3 and R4 form, with the nitrogen atom which bears them, a heterocyclic group comprising 3 to 7 ring members that may incorporate an oxygen or sulphur atom, an NR group or an NR'-CO group, wherein said ring is optionally substituted with one or more groups selected from a halogen atom or a (C1-C6)alkyl, (C1-C6)alkoxy, halo(C1-C6)alkyl or halo(C1- C6)alkoxy group, R2 is an aryl group, optionally substituted with one or more groups selected from a halogen atom or a methyl, trifluoromethyl, methoxy or trifluoromethoxy group. Process for the preparation thereof and therapeutic use thereof.
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