发明名称 |
PROTEIN KINASE INHIBITORS AND METHODS FOR USING THEREOF |
摘要 |
<p>The invention provides compounds of formula (l) and pharmaceutical compositions thereof, which are useful as protein kinase inhibitors, and methods for using such compounds to treat, ameliorate or prevent a condition associated with abnormal or deregulated kinase activity. In some embodiments, the invention provides methods for using such compounds to treat, ameliorate or prevent diseases or disorders that involve abnormal activation of AIk, AbI, Aurora-A, B-Raf, C-Raf, Bcr-Abl, BRK, BIk, Bmx, BTK, c-Kit, c-RAF, CSK, c-SRC, EphBl, EphB2, EphB4, FLTl, Fms, Flt3, Fyn, FRK3, JAK2, KDR, Lck, Lyn, PDGFRalpha, PDGFRbeta, PKCalpha, SAPK2alpha, Src, SIK, Syk, Tie2 and TrkB kinases.</p> |
申请公布号 |
WO2008144253(A1) |
申请公布日期 |
2008.11.27 |
申请号 |
WO2008US63187 |
申请日期 |
2008.05.09 |
申请人 |
IRM LLC;REN, PINGDA;WANG, XIA;JIANG, SONGCHUN;NAGLE, ADVAIT;OKRAM, BARUN;HE, YUN;XIE, YONGPING;WANG, XING;HUANG, SHENLIN;WANG, XIAODONG;LIU, YI;ALBAUGH, PAMELA, A.;GRAY, NATHANAEL, S.;ZHANG, GUOBAO |
发明人 |
REN, PINGDA;WANG, XIA;JIANG, SONGCHUN;NAGLE, ADVAIT;OKRAM, BARUN;HE, YUN;XIE, YONGPING;WANG, XING;HUANG, SHENLIN;WANG, XIAODONG;LIU, YI;ALBAUGH, PAMELA, A.;GRAY, NATHANAEL, S.;ZHANG, GUOBAO |
分类号 |
C07D471/04;A61K31/519;A61P35/00;C07D487/04 |
主分类号 |
C07D471/04 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|