发明名称 Pyridyl acetic acid compounds
摘要 The present invention provides a compound represented by the formula (I): wherein R1 is a C?1-6#191 alkyl group optionally substituted by a C?3-10#191 cycloalkyl group, R2 is a C?2-6#191 alkyl group, R3 is a hydrogen atom, a C?1-6#191 alkyl group or a halogen atom, and X is -OR6 or -NR4R5 wherein R4 and R6 are each independently a hydrogen atom, an optionally substituted hydrocarbon group or an optionally substituted heterocyclic group, R5 is an optionally substituted hydrocarbon group, an optionally substituted heterocyclic group or an optionally substituted hydroxy group, or R4 and R5 optionally form, together with the adjacent nitrogen atom, an optionally substituted nitrogen-containing heterocycle, or a salt thereof. The compound of the present invention has a superior peptidase inhibitory action and is useful as an agent for the prophylaxis or treatment of diabetes and the like.
申请公布号 ZA200708144(B) 申请公布日期 2008.11.26
申请号 ZA20070008144 申请日期 2006.02.24
申请人 TAKEDA PHARMACEUTICAL COMPANY LIMITED 发明人 MAEZAKI, HIRONOBU;SUZUKI, NOBUHIRO
分类号 A61K;A61P;C07D 主分类号 A61K
代理机构 代理人
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