发明名称 Amino-5-(6-membered)heteroarylimidazolone compounds and the use thereof for beta-secretase modulation
摘要 The present invention provides a 2-amino-5-heteroaryl-5-phenylimidazolone compound of formula I The present invention also provides methods for the use thereof to inhibit beta-secretase (BACE) and treat beta-amyloid deposits and neurofibrillary tangles.
申请公布号 US7452885(B2) 申请公布日期 2008.11.18
申请号 US20060478098 申请日期 2006.06.29
申请人 WYETH 发明人 ZHOU PING;MALAMAS MICHAEL SOTIRIOS;LI YANFANG;ROBICHAUD ALBERT JEAN;QUAGLIATO DOMINICK ANTHONY
分类号 C07D403/04;A61K31/4439 主分类号 C07D403/04
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